Orlistat Cas: 96829-58-2
| Catalog Number | xwm 91190 |
| Khoom npe | Orlistat |
| CAS | 96829-58-2 |
| Molecular Formula | C29H53 NPO 5 |
| Molecular Luj | 495.73 ib |
| Cov ntaub ntawv khaws cia | 2 txog 8 ° C |
Khoom Specification
| Qhov tshwm sim | Dawb hmoov |
| Assay | 99% |
Cov tshuaj poob phaus thiab lipid-txo cov tshuaj tshiab: Orlistat yog ib yam tshiab ntawm kev poob phaus thiab lipid-txo cov tshuaj tam sim no thoob ntiaj teb lees paub.Nrog rau kev muag khoom txhua xyoo ntawm US $ 538 lab, orlistat tam sim no nyob 80% ntawm lub ntiaj teb poob kev lag luam, thiab kev muag khoom txhua xyoo hauv Hong Kong, Tuam Tshoj ib leeg ncav cuag US $ 80 lab.Tam sim no nws tsuas yog OTC cov tshuaj poob phaus hauv ntiaj teb.Ntau tshaj 40,000,000 tus neeg thoob ntiaj teb tau noj nws thiab ua tiav qhov hnyav.Tam sim no nws yog qhov zoo tshaj plaws-muag khoom poob phaus.Nws muaj txiaj ntsig zoo rau kev poob phaus.Orlistat yog ib qho muaj zog thiab ua haujlwm ntev ntev ntawm lub plab hnyuv lipase inhibitor.Los ntawm ncaj qha thaiv lub cev nqus cov rog hauv cov zaub mov, thaum noj cov calories thiab rog tsawg dua li kev noj, Lub cev rog yog ib txwm txo qis, thiaj li ua tiav lub hom phiaj ntawm kev poob phaus.Nws muaj kev nyab xeeb kom poob phaus, cov khoom xyaw nquag tsis nkag mus rau hauv cov ntshav ncig, thiab tsis ua rau lub hauv nruab nrab lub paj hlwb.
Orlistat yog ib qho kev ua haujlwm ntev thiab muaj zog tshwj xeeb hauv plab hnyuv lipase inhibitor, hmoov dawb lossis dawb dawb ntawm chav sov, tsis muaj dej, soluble hauv chloroform, thiab yooj yim soluble hauv ethanol.Lub active serine chaw ntawm gastric lipase thiab pancreatic lipase tsim covalent bonds kom inactivate cov enzymes.Cov rog hauv cov zaub mov tsis tuaj yeem decomposed rau hauv cov rog dawb thiab monoacylglycerols, yog li cov rog tsis tuaj yeem nqus tau thiab siv, yog li txo lub cev calorie kom tsawg thiab tswj lub cev hnyav.Cov tshuaj no tsis tas yuav muaj kev nqus dej ua haujlwm.Ntawm cov koob tshuaj ib txwm muaj, qhov nqus ntawm cov rog tuaj yeem cuam tshuam los ntawm 30%.Nws tsis tshua muaj txiaj ntsig tom qab kev tswj hwm qhov ncauj, thiab tuaj yeem cuam tshuam los ntawm cov metabolism hauv cov hnyuv.Qhov chaw metabolic yog nyob rau hauv cov phab ntsa ntawm txoj hnyuv, thiab kev tshem tawm ib nrab ntawm lub neej yog li 14 mus rau 19 teev.Kwv yees li 97% ntawm cov khoom no tau tawm nrog cov quav, ntawm 83% yog tawm hauv nws daim ntawv qub.
Nws tuaj yeem siv rau hauv kev kho mob rog rog thiab hyperlipidemia.Raws li ib txwm muaj, koob tshuaj 120 mg tuaj yeem noj hauv qhov ncauj, peb zaug hauv ib hnub, nrog zaub mov lossis 1 teev tom qab noj mov.Qhov hnyav tuaj yeem pib poob tom qab 2 lub lis piam ntawm kev noj tshuaj.Nws tuaj yeem noj tsis tu ncua rau 6 txog 12 lub hlis.Yog tias qhov koob tshuaj tau nce mus rau ntau dua 400 mg ib hnub, nws cov nyhuv yuav tsis raug kho ntxiv lawm.
